Dostinex (Cabergoline)
Dostinex, containing the active ingredient Cabergoline, is a dopamine receptor agonist medication used primarily to treat hyperprolactinemia – a condition characterized by abnormally high levels of prolactin hormone. This prolactin inhibitor helps reduce the levels of the hormone in the blood, leading to a normalization of menstrual cycles, improved fertility, and relief from other symptoms associated with high prolactin.
Why Choose Dostinex (Cabergoline)?
- Effective Prolactin Reduction: Dostinex effectively lowers elevated prolactin levels, helping restore hormonal balance.
- Improved Fertility and Menstrual Regularity: Helps regulate ovulation and menstrual cycles in women affected by hyperprolactinemia.
- Minimal Dosing Frequency: Taken only twice a week due to its long-lasting action.
- Well-Tolerated Formula: Generally well-tolerated by most patients, ensuring effective treatment with minimal side effects.
How to Use Dostinex (Cabergoline)?
- Starting Dose: 0.25 mg twice a week.
- Maintenance Dose: The dosage can be adjusted based on the patient’s prolactin levels, typically ranging from 0.25 mg to 1 mg twice a week.
- Maximum Dose: Should not exceed 3 mg per week.
- Can be taken with or without food.
- Swallow tablets whole with water.
- Regular monitoring of prolactin levels is recommended for optimal dosing.
Important Safety Information about Dostinex
- Regular cardiovascular assessment is recommended due to the potential risk of valvulopathy.
- Use with caution in patients with cardiovascular disease or severe renal impairment.
- Inform your healthcare provider of all medications you’re taking to avoid potential drug interactions.
- Store at room temperature (15°C to 25°C).
- Keep in a dry place, away from moisture and direct sunlight.
- Keep out of reach of children.
Fact Table for Dostinex
| Facts | Details |
| Generic Name | Cabergoline |
| Brand Names | Dostinex |
| Drug Class | Dopamine agonist |
| FDA Approval | Approved by the FDA in 1996 |
| Indications | Primarily used to treat disorders associated with high levels of prolactin (hyperprolactinemia) |
| Mechanism of Action | Works by mimicking the activity of dopamine, a substance in the brain that helps control mood and behavior, thus decreasing the production of prolactin by the pituitary gland |
| Dosage Forms | Oral tablets |
| Common Dosage | Typically starts at 0.25 mg twice weekly, adjusted according to patient response and prolactin levels |
| Side Effects | Nausea, headache, dizziness, fatigue, dry mouth, constipation, depression, hypotension |
| Contraindications | Uncontrolled hypertension, history of cardiac valvulopathy, fibrotic disorders |
| Drug Interactions | Can interact with other dopamine antagonists, certain antipsychotics, and antiemetics |
| Pregnancy Category | Category B (No evidence of risk in humans, but studies are limited) |
| Breastfeeding | Not recommended as it may inhibit lactation and/or pass into breast milk |
| Monitoring Requirements | Regular monitoring of heart function and prolactin levels is necessary |
Common Side Effects of Dostinex
Like all medications, Dostinex (Cabergoline) can cause side effects, although not everybody gets them. Understanding these side effects can help you use this medication safely and effectively.
- Nausea
- Headache
- Dizziness
- Fatigue
- Dry mouth
If you experience any side effects, discuss them with your healthcare provider. They can offer advice and may adjust your treatment if necessary. Report any severe or unexpected side effects immediately.
How Can You Buy Dostinex (Cabergoline)?
You can order Dostinex (Cabergoline) using these methods on our website:
- Order Online
- Order by Phone
- Order by Fax
- Order your refills
Visit our How to order page.
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He supports other members of the healthcare team including physicians, mid-level providers, nurses, and other clinical staff.
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